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Journal articles
Fluoroazaindolines by an uncommon radical ipso-substitution of a C-F bond
Abstract : Trifluoroazaindoline derivatives are prepared using the first synthetically useful radical ipso-substitution of a fluorine atom. The initial procedure has been improved to allow the gram scale synthesis of these building blocks, which can be regioselectively substituted by nucleophiles under mild conditions to rapidly access a library of new molecules. Oxidation to the corresponding fluoroazaindole core has also been accomplished. © 2011 CSIRO.
https://hal-polytechnique.archives-ouvertes.fr/hal-00950022
Contributor : Denis Roura <>
Submitted on : Wednesday, February 26, 2014 - 9:49:44 AM
Last modification on : Thursday, March 5, 2020 - 6:25:14 PM
Contributor : Denis Roura <>
Submitted on : Wednesday, February 26, 2014 - 9:49:44 AM
Last modification on : Thursday, March 5, 2020 - 6:25:14 PM