Au-Catalyzed Formation of Functionalized Quinolines from 2-Alkynyl Alkyl Azides Derivatives

Colombe Gronnier; Guillaume Boissonnat; Fabien Gagosz

doi:10.1021/ol4019634

Journal articles

Au-Catalyzed Formation of Functionalized Quinolines from 2-Alkynyl Alkyl Azides Derivatives

Colombe Gronnier ¹ Guillaume Boissonnat ¹ Fabien Gagosz ¹

1 DCSO - Laboratoire de synthèse organique

Abstract : A new method for converting 2-alkynyl arylazide derivatives into functionalized polysubstituted quinolines following a gold-catalyzed 1,3-acetoxy shift/cyclization/1,2-group shift sequence has been developed. This transformation proceeds under mild reaction conditions, is efficient, and tolerates a large variety of functional groups.

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Submitted on : Wednesday, March 26, 2014 - 9:46:28 PM
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Au-Catalyzed Formation of Functionalized Quinolines from 2-Alkynyl Alkyl Azides Derivatives

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Au-Catalyzed Formation of Functionalized Quinolines from 2-Alkynyl Alkyl Azides Derivatives

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