A convergent route to functional protected amines, diamines, and β-amino acids

Abstract : Phthalimide protected amines react with NBS under peroxide initiation to give geminal phthalimido-bromo derivatives, which are readily converted into the corresponding xanthates. These xanthates in turn undergo radical additions to numerous olefins, providing a convergent and modular access to densely functionalized protected amines and diamines.
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Tetrahedron, Elsevier, 2014, 70 (40), pp.7192-7206. 〈10.1016/j.tet.2014.07.055〉
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https://hal-polytechnique.archives-ouvertes.fr/hal-01082412
Contributeur : Denis Roura <>
Soumis le : jeudi 13 novembre 2014 - 14:32:11
Dernière modification le : jeudi 10 mai 2018 - 02:07:51

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Songzhe Han, Rachel A. Jones, Béatrice Quiclet-Sire, Samir Z. Zard. A convergent route to functional protected amines, diamines, and β-amino acids. Tetrahedron, Elsevier, 2014, 70 (40), pp.7192-7206. 〈10.1016/j.tet.2014.07.055〉. 〈hal-01082412〉

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